Drug | MBD3L2 EC50 (nanomolar) | MYH2 EC50 (nanomolar) | Mechanism |
---|---|---|---|
Clenbuterol hydrochloride | <Â 60 | >Â 5000 | Beta-2 adrenergic agonist |
Tulobuterol hydrochloride | <Â 60 | >Â 5000 | Beta-2 adrenergic agonist |
Albuterol | <Â 60 | <Â 60 | Beta-2 adrenergic agonist |
Fenoterol hydrobromide | <Â 60 | <Â 60e | Beta-2 adrenergic agonist |
Fluticasone | <Â 60 | <Â 60d | Glucocorticoid |
Nylidrin (Buphenine isoxsuprine) | <Â 60 | <Â 60c | Beta-2 adrenergic agonist |
Sirolimus | <Â 60 | <Â 60 | Immunosuppressant |
Terbutaline hemisulfate | <Â 60 | <Â 60c | Beta-2 adrenergic agonist |
Vinblastine | <Â 60b | <Â 60 | Antineoplastic, spindle poison |
Dequalinium | 70 | 5000 | Anti-infective, antineoplastic |
Bisoctrizole | 100c | >Â 5000 | Sunscreen |
Isoetharine | 100 | 5000 | Beta-1 and beta-2 adrenergic agonist |
Penicillamine | 180c | >Â 5000 | Chelating agent |
Benzethonium chloride | 190 | 400 | Anti-infective |
Cetylpyridinium chloride | 200 | 300 | Anti-infective |
Epinephrine bitartrate | 200 | 4000 | Alpha and beta-adrenergic agonist |
Phenylephrine | 200 | 4000 | Alpha-1 adrenergic agonist |
Piromidic acid | <Â 500a | >Â 5000 | Antibacterial |
Acenocoumarol | 500b | >Â 5000 | Anticoagulant |
Atorvastatin | 500c | >Â 5000 | HmG-CoA reductase inhibitor |
Cresopirine | 500 | >Â 5000 | Anti-inflammatory, fever reducer |
Dicoumarol | 500b | >Â 5000 | Anticoagulant |
Thiostrepton | 500 | 700f | Antibacterial |
Thimerosal | 500 | Â | Anti-infective, organomercury |
Ethylnorepinephrine | 600 | 5000 | Alpha and beta adrenergic agonist |
Fluvoxamine | 1000 | 4000 | SSRI, antidepressant |
Clozapine | 1000 | 2000 | Antipsychotic |
Adrenalone hydrochloride | 1000 | 1500 | Alpha-adrenergic agonist |
Butamben | 1000f | 1000 | Local anesthetic |
Thonzonium | 1000 | 1000 | Mucolytic antibacterial |
Mebendazole | 1000f | Â | Anthelmintic |
Puromycin | 1000f | Â | Antibacterial, antineoplastic |
Colforsin | 1500d | >Â 5000 | Adenylyl cyclase activator |
Dimercaprol | 1500 | 3000 | Chelating agent |
Benzalkonium | 1500 | Â | Anti-infective |
Norepinephrine | 1600 | 4000 | Alpha and beta adrenergic agonist |
Polymyxin B | 1700 | 3500 | Antibacterial |
Oxedrine (synephrine) | 2000 | 5000 | Alpha and beta adrenergic agonist and antagonist |
Nonoxynol-9 | 2000 | Â | Spermicide |
Papaverine | 2500 | 10,000 | Vasodilator |
Pentamidine | 3000 | Â | Antiprotozoal |
Triamcinolone | 3000 | Â | Corticosteroid |
Dichlorephen | 3500 | Â | Anthelmintic |
Ebselen | 4000 | Â | Antioxidant, anti-inflammatory |
Minocycline | 5000 | 10,000 | Antibacterial |
Inosine | 5000 | >Â 5000 | Nucleoside |
Sulbentine | 5000 | >Â 5000 | Antifungal |
Artesunate | 5000 | Â | Anti-malarial |
Broxaldine | 5000 | Â | Antifungal |
Broxyquinoline | 5000 | Â | Anti-infectant |
Meclocycline | 5000 | Â | Antibacterial |
Sennoside A | 5000 | Â | Cathartic/laxative |