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Table 1 Cayman chemical epigenetics screening library

From: A novel chemical-combination screen in zebrafish identifies epigenetic small molecule candidates for the treatment of Duchenne muscular dystrophy

Plate 1

Plate 2

Well

Small molecule

Well

Small molecule

A2

3-amino benzamide

A2

AGK2

A3

SB 939

A3

CAY10603

A4

PCI 34051

A4

Chaetocin

A5

4-iodo-SAHA

A5

Splitomicin

A6

Sirtinol

A6

CBHA

A7

C646

A7

M 344

A8

Ellagic acid

A8

Oxamflatin

A9

Scriptaid

A9

Salermide

A10

Suberohydroxamic acid

A10

Mirin

A11

Apicidin

A11

Pimelic diphenylamide 106

B2

UNC0321 (trifluoroacetate salt)

B2

(S)-HDAC-42

B3

(−)-Neplanocin A

B3

MS-275

B4

Cl-Amidine

B4

HNHA

B5

F-Amidine (trifluoroacetate salt)

B5

RG-108

B6

JGB1741

B6

2′,3′,5′-triacetyl-5-azacytidine

B7

UNC0638

B7

S-Adenosylhomocysteine

B8

Phthalazinone pyrazole

B8

UNC0224

B9

Isoliquiritigenin

B9

Chidamide

B10

CCG-100602

B10

3-Deazaneplanocin A

B11

CAY10669

B11

Sinefungin

C2

Zebularine

C2

Pyroxamide

C3

Delphinidin chloride

C3

WDR5-0103

C4

ITF 2357

C4

AMI-1 (sodium salt)

C5

PFI-1

C5

UNC1215

C6

5-Azacytidine

C6

GSK 343

C7

Decitabine

C7

SIRT1/2 inhibitor IV

C8

(+)-JQ1

C8

I-CBP112 (hydrochloride)

C9

(−)-JQ1

C9

UNC1999

C10

BSI-201

C10

PFI-3

C11

1-Naphthoic acid

C11

trans-Resveratrol

D2

Sodium 4-phenylbutyrate

D2

2,4-DPD

D3

IOX1

D3

DMOG

D4

MI-2 (hydrochloride)

D4

Trichostatin A

D5

MI-nc (hydrochloride)

D5

CAY10398

D6

Gemcitabine

D6

RSC-133

D7

Lomeguatrib

D7

KD 5170

D8

Octyl-α-ketoglutarate

D8

CAY10433

D9

Daminozide

D9

Piceatannol

D10

GSK-J1 (sodium salt)

D10

CAY10591

D11

GSK-J2 (sodium salt)

D11

EX-527

E2

GSK-J4 (hydrochloride)

E2

SAHA

E3

GSK-J5 (hydrochloride)

E3

2-PCPA (hydrochloride)

E4

CPTH2

E4

Nicotinamide

E5

Valproic acid (sodium salt)

E5

BIX01294

E6

Tenovin-1

E6

N-Oxalylglycine

E7

Tenovin-6

E7

Suramin (sodium salt)

E8

Sodium butyrate

 

E9

Anacardic acid

 
  1. The identities of the chemicals and composition of the library, 94 chemicals distributed over two 96-well plates, are shown. The library (Cayman Chemical Item No. 11076, Batch No. 0455098) was received as 10 mM stocks of each chemical in DMSO