Compound | % inhibition of ZSCAN4 reporter | % inhibition of Renilla luciferase | Mechanism |
---|---|---|---|
(+)-JQ1 | 99 (1 μMa) | 27 (1 μMa) | BET bromodomain inhibitor |
PFI-1 | 89 (1 μMa) | 0 (1 μMa) | BET bromodomain inhibitor |
SGC-CBP30 | 75 (1 μMa) | 24 (1 μMa) | CBP/p300 bromodomain inhibitor |
Bromosporine | 92 (2 μMa) | 9 (2 μMa) | Pan-bromodomain inhibitor |